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Study breakdown

Surprising: GHRH Can Also Activate the Ghrelin Receptor

In VitroModerate evidence
The takeaway

GHRH (growth hormone-releasing hormone) unexpectedly activated the GHS-R1a (ghrelin receptor), revealing cross-talk between the two GH-releasing receptor systems that were thought to be completely independent.

Key finding

GHRH demonstrated agonist activity at the GHS-R1a (ghrelin receptor) at physiologically relevant concentrations, revealing previously unknown cross-ta

What the researchers found

GHRH demonstrated agonist activity at the GHS-R1a (ghrelin receptor) at physiologically relevant concentrations, revealing previously unknown cross-talk between the GHRH and ghrelin receptor systems — explaining some synergistic GH-releasing effects.

Why it matters

Relevant for ghrp, cjc-1295, receptor-signaling.

How the study worked

in-vitro study.

What this study cannot tell us

See abstract.

How to read the evidence

moderate evidence.

When this study was published

Published in 2008.

The bigger picture

Advances peptide research.

Questions still open

  • Further research needed.
  • Clinical translation to evaluate.

Common questions

What was studied?
Surprising: GHRH Can Also Activate the Ghrelin Receptor
What was found?
GHRH (growth hormone-releasing hormone) unexpectedly activated the GHS-R1a (ghrelin receptor), revealing cross-talk between the two GH-releasing receptor systems that were thought to be completely independent.

Read the original research

Growth hormone-releasing hormone as an agonist of the ghrelin receptor GHS-R1a.

Proceedings of the National Academy of Sciences of the United States of America, 105(51), 20452-7

Citation

Casanueva, Felipe F; Camiña, Jesus P; Carreira, Marcos C; Pazos, Yolanda; Varga, Jozsef L; Schally, Andrew V. (2008). Growth hormone-releasing hormone as an agonist of the ghrelin receptor GHS-R1a.. Proceedings of the National Academy of Sciences of the United States of America, 105(51), 20452-7. https://doi.org/10.1073/pnas.0811680106