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Study breakdown

Anti-CGRP drugs reduce cortical hyperexcitability in migraine responders as shown by functional brain imaging

evidence
The takeaway

In 36 migraine patients, galcanezumab responders (≥50% MMD reduction) showed reduced resting-state functional connectivity between somatosensory, motor, insular, and visual cortices after 3 months, while non-responders showed no changes.

Brain rewiring in responders

Anti-CGRP therapy reduced cortical hyperexcitability in migraine responders—the first fMRI evidence of brain connectivity normalization from neuropeptide-targeted treatment

What the researchers found

Responders (19/36): ↓functional connectivity between somatosensory/motor cortex, insula, and visual areas. Non-responders (17/36): no changes. No baseline differences between groups. 3-month galcanezumab treatment.

Why it matters

This provides the first neuroimaging evidence of how anti-CGRP drugs change brain function. Reducing cortical hyperexcitability explains the clinical benefit and suggests CGRP blockade initiates neural recovery beyond just pain relief.

How the study worked

Prospective resting-state fMRI study. 36 patients (high-frequency EM or CM). Pre- and post-3-month galcanezumab. ROI-to-ROI connectivity analysis. Responder (≥50% MMD reduction) vs non-responder comparison.

What this study cannot tell us

Small sample (36). Cannot determine if brain changes cause or result from clinical improvement. 3-month follow-up is short. Galcanezumab only—other CGRP drugs may differ.

How to read the evidence

Prospective neuroimaging study with responder/non-responder comparison. Good mechanistic evidence but small sample.

When this study was published

Published in 2025.

The bigger picture

Migraine is increasingly understood as a brain connectivity disorder. This study shows anti-CGRP drugs can normalize cortical communication patterns, providing neurobiological evidence for disease modification rather than just symptom relief.

Questions still open

  • Do brain connectivity changes persist after stopping CGRP therapy?
  • Could baseline fMRI predict who will respond to anti-CGRP drugs?
  • Do the connectivity changes progress with longer treatment?

Common questions

Do anti-CGRP drugs change the brain?
Yes. This imaging study showed that migraine patients who responded to galcanezumab had measurable changes in brain connectivity after 3 months—reduced communication between pain-processing, sensory, and visual areas. This suggests the brain's hyperexcitable state in migraine normalizes when CGRP signaling is blocked.
What does this mean for migraine treatment?
It suggests anti-CGRP drugs do more than just relieve individual migraine attacks—they may actually shift the brain from a migraine-prone state to a more normal state. Non-responders showed no brain changes, which could help explain why some patients benefit while others do not.

Read the original research

Peripherally acting anti-CGRP monoclonal antibodies attenuate cortical resting-state connectivity in migraine patients.

Cephalalgia : an international journal of headache, 45(2), 3331024241313377

Citation

Szabo, Edina; Bolo, Nicolas R; Borsook, David; Burstein, Rami; Ashina, Sait. (2025). Peripherally acting anti-CGRP monoclonal antibodies attenuate cortical resting-state connectivity in migraine patients.. Cephalalgia : an international journal of headache, 45(2), 3331024241313377. https://doi.org/10.1177/03331024241313377