Neuropeptide Y offers a new biological target for treatment-resistant depression through stress and inflammation pathways

Decreased cerebrospinal NPY levels and altered hippocampal NPY receptor expression in treatment-resistant depression patients suggest NPY restoration—via intranasal delivery or receptor-selective modulation—as a novel therapeutic approach.

Singanwad, Priyanka et al.·Neuropeptides·2025·
RPEP-136112025RETHINKTHC RESEARCH DATABASErethinkthc.com/research

Quick Facts

Study Type
Not classified
Evidence
Not graded
Sample
Not reported

What This Study Found

Decreased CSF NPY in TRD patients. Reduced NPY receptor expression in stress-related brain regions. Animal models: NPY dysregulation in chronic stress with altered hippocampal signaling and HPA axis. Therapeutic targets: intranasal NPY, receptor-selective modulators.

Key Numbers

How They Did This

Narrative review synthesizing preclinical (animal stress models) and clinical (CSF biomarker, receptor expression) evidence for NPY in TRD.

Why This Research Matters

TRD affects about one-third of depressed patients and has few effective treatments. NPY represents a biologically grounded target distinct from serotonin/norepinephrine pathways targeted by conventional antidepressants.

The Bigger Picture

Moving beyond serotonin-based depression treatment toward neuropeptide targets could transform mental health care. NPY's involvement in stress, inflammation, and neuroplasticity makes it a uniquely comprehensive target for treatment-resistant cases.

What This Study Doesn't Tell Us

Review format. Clinical NPY data limited. Intranasal NPY delivery still experimental. Causation vs association for NPY decreases in TRD unclear.

Questions This Raises

  • ?Will intranasal NPY clinical trials show efficacy for TRD?
  • ?Which NPY receptor subtype is most important for antidepressant effects?
  • ?Could NPY levels serve as biomarkers to predict TRD?

Trust & Context

Key Stat:
NPY depleted in TRD Decreased cerebrospinal NPY and reduced receptor expression in stress-related brain regions suggest NPY restoration as a novel antidepressant strategy
Evidence Grade:
Review of preclinical and clinical evidence. Good biological rationale but therapeutic applications are still experimental.
Study Age:
Published in 2025.
Original Title:
Neuropeptide Y as a multifaceted modulator of neuroplasticity, Neuroinflammation, and HPA axis dysregulation: Perceptions into treatment-resistant depression.
Published In:
Neuropeptides, 112, 102538 (2025)
Database ID:
RPEP-13611

Evidence Hierarchy

Meta-Analysis / Systematic Review
Randomized Controlled Trial
Cohort / Case-Control
Cross-Sectional / ObservationalSnapshot without intervening
This study
Case Report / Animal Study
What do these levels mean? →

Frequently Asked Questions

What is treatment-resistant depression?

TRD is depression that does not improve with standard antidepressant medications (typically after trying 2+ drugs). It affects about one-third of depressed patients and is a major unmet medical need. This review identifies neuropeptide Y as a potential new treatment target.

How could NPY help depression?

NPY regulates stress responses, inflammation, and brain plasticity—all disrupted in depression. People with TRD have lower NPY levels in their brain fluid. Restoring NPY through nasal spray delivery or drugs that activate NPY receptors could address depression through fundamentally different mechanisms than current antidepressants.

Read More on RethinkPeptides

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Cite This Study

RPEP-13611·https://rethinkpeptides.com/research/RPEP-13611

APA

Singanwad, Priyanka; Tatode, Amol; Qutub, Mohammad; Taksande, Brijesh; Umekar, Milind; Trivedi, Rashmi; Premchandani, Tanvi. (2025). Neuropeptide Y as a multifaceted modulator of neuroplasticity, Neuroinflammation, and HPA axis dysregulation: Perceptions into treatment-resistant depression.. Neuropeptides, 112, 102538. https://doi.org/10.1016/j.npep.2025.102538

MLA

Singanwad, Priyanka, et al. "Neuropeptide Y as a multifaceted modulator of neuroplasticity, Neuroinflammation, and HPA axis dysregulation: Perceptions into treatment-resistant depression.." Neuropeptides, 2025. https://doi.org/10.1016/j.npep.2025.102538

RethinkPeptides

RethinkPeptides Research Database. "Neuropeptide Y as a multifaceted modulator of neuroplasticit..." RPEP-13611. Retrieved from https://rethinkpeptides.com/research/singanwad-2025-neuropeptide-y-as-a

Access the Original Study

Study data sourced from PubMed, a service of the U.S. National Library of Medicine, National Institutes of Health.

This study breakdown was produced by the RethinkPeptides research team. We analyze and report published research findings without making health recommendations. All interpretations are based solely on the published abstract and study data.