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Research citation

Formulation of pH-responsive nanoplexes based on an antimicrobial peptide and sodium alginate for targeted delivery of vancomycin against resistant bacteria.

Laboratory And Animal StudyPreliminary evidence

This record provides bibliographic details and links to the original research. An editorial study breakdown is not available.

What the researchers found

pH-responsive nanoplexes combining a plant antimicrobial peptide with vancomycin showed 2-fold stronger activity against MRSA, 5-fold better biofilm eradication, and 4-5 fold reduced bacterial burden in kidneys, liver, and blood of mice with MRSA infection.

Why it matters

MRSA is a leading cause of hospital deaths. This nanoparticle delivery system makes vancomycin far more effective by combining it with an antimicrobial peptide in a pH-triggered release system.

The numbers in context

Particle size 159.5 nm. Encapsulation efficiency 82.34%. 2-fold enhanced activity vs S. aureus and MRSA. 5-fold greater MRSA biofilm eradication. In vivo: 5-fold reduction in kidney MRSA, 4-fold in liver and blood. pH-accelerated VCM release at acidic pH.

How the study worked

Formulated nanoplexes from plant AMP and sodium alginate loaded with vancomycin. Characterized size, zeta potential, encapsulation, pH-responsive release. In vitro: MIC, biofilm eradication. In vivo: MRSA systemic infection in mice, organ bacterial burden, inflammation markers.

Who was studied

Mice with MRSA systemic infection; S. aureus and MRSA in vitro

What this study cannot tell us

Specific plant AMP not named in abstract. Mouse model may not reflect human MRSA infection. Toxicity profile needs more characterization. Manufacturing scalability not addressed.

Read the original research

Formulation of pH-responsive nanoplexes based on an antimicrobial peptide and sodium alginate for targeted delivery of vancomycin against resistant bacteria.

Biological chemistry, 406(8-9), 369-389

Citation

Shahin, Shourok; Omolo, Calvin A; Elhassan, Eman; Ismail, Eman A; Farukh, Sania; Govender, Jasoda; Faya, Mbuso; Govender, Thirumala. (2025). Formulation of pH-responsive nanoplexes based on an antimicrobial peptide and sodium alginate for targeted delivery of vancomycin against resistant bacteria.. Biological chemistry, 406(8-9), 369-389. https://doi.org/10.1515/hsz-2025-0142