Amylin receptors as therapeutic targets in obesity: Emerging peptide-based strategies.

Rejili, Mokhtar et al.·Vascular pharmacology·2025·Moderate EvidenceReview
RPEP-13237ReviewModerate Evidence2025RETHINKTHC RESEARCH DATABASErethinkthc.com/research

Quick Facts

Study Type
Review
Evidence
Moderate Evidence
Sample
N=Not applicable (review)
Participants
Adults with obesity (focus of reviewed therapies)

What This Study Found

Amylin receptor agonists like cagrilintide and dual-action compounds show strong potential for obesity treatment, especially when combined with GLP-1 receptor agonists, by targeting both homeostatic and reward-driven eating pathways.

Key Numbers

Not specified in abstract. References pramlintide, cagrilintide, KBP-series DACRAs, ZP8396, and amycretin.

How They Did This

Narrative review of preclinical and clinical evidence on amylin receptor agonists for obesity. Covers molecular pharmacology, clinical development, genetic variants, and combination strategies.

Why This Research Matters

GLP-1 drugs alone produce meaningful but limited weight loss. Adding amylin-based drugs could push results further by targeting a different hormone system that controls hunger, stomach emptying, and food reward.

What This Study Doesn't Tell Us

Narrative review without systematic search or meta-analysis. Most amylin-based agents are still investigational. Long-term efficacy and safety data are limited. Disease-modifying effects beyond weight loss remain unproven.

Trust & Context

Original Title:
Amylin receptors as therapeutic targets in obesity: Emerging peptide-based strategies.
Published In:
Vascular pharmacology, 162, 107563 (2025)
Database ID:
RPEP-13237

Evidence Hierarchy

Meta-Analysis / Systematic Review
Randomized Controlled Trial
Cohort / Case-Control
Cross-Sectional / ObservationalSnapshot without intervening
This study
Case Report / Animal Study

Summarizes existing research on a topic.

What do these levels mean? →

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Cite This Study

RPEP-13237·https://rethinkpeptides.com/research/RPEP-13237

APA

Rejili, Mokhtar; Hussain, Md Sadique; Khan, Yumna; Haouala, Faouzi; Ganesan, Subbulakshmi; Sahoo, Samir; Pal, Amrita; Arora, Vimal. (2025). Amylin receptors as therapeutic targets in obesity: Emerging peptide-based strategies.. Vascular pharmacology, 162, 107563. https://doi.org/10.1016/j.vph.2025.107563

MLA

Rejili, Mokhtar, et al. "Amylin receptors as therapeutic targets in obesity: Emerging peptide-based strategies.." Vascular pharmacology, 2025. https://doi.org/10.1016/j.vph.2025.107563

RethinkPeptides

RethinkPeptides Research Database. "Amylin receptors as therapeutic targets in obesity: Emerging..." RPEP-13237. Retrieved from https://rethinkpeptides.com/research/rejili-2025-amylin-receptors-as-therapeutic

Access the Original Study

Study data sourced from PubMed, a service of the U.S. National Library of Medicine, National Institutes of Health.

This study breakdown was produced by the RethinkPeptides research team. We analyze and report published research findings without making health recommendations. All interpretations are based solely on the published abstract and study data.