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Study breakdown

Platelets have renin-angiotensin system receptors but angiotensin peptides do not affect platelet function

In VitroLow evidence
The takeaway

Although human platelets express all major renin-angiotensin system receptors, angiotensin peptides did not influence platelet adhesion or aggregation, suggesting COVID-19 coagulopathy may not be driven by RAS-platelet interactions.

Expressed but inactive

All six RAS receptors present on platelets, but no angiotensin peptide affected platelet function at any concentration

What the researchers found

Healthy human platelets express RAS receptors (Mas, MrgD, ACE, ACE2, AT1, AT2) but angiotensin peptides (Ang-I, Ang-II, Ang-(1-7), Ang-(1-9), alamandine) had no effect on platelet adhesion or aggregation at any concentration tested. ACE activity was present but captopril-resistant; ACE2 was undetectable.

Why it matters

This negative finding is important because it helps rule out direct RAS-platelet interactions as a mechanism for COVID-19 coagulopathy, redirecting research toward other pathways. It also clarifies the functional status of RAS components in platelets.

The numbers in context

Tested Captopril, Alamandine, Angiotensin-I, Angiotensin-II, Angiotensin-(1-7), and Angiotensin-(1-9) across a wide range of concentrations. Measured adhesion by BCECF fluorescence and aggregation by aggregometry.

How the study worked

Ex vivo study on healthy human platelets using western blot and immunofluorescence for receptor expression, spectrophotometry for adhesion, aggregometry for activation/aggregation, and fluorescent peptide substrates for enzyme activity.

Who was studied

Healthy human platelet samples (ex vivo)

What this study cannot tell us

Study used only healthy donor platelets—results may differ in disease states (COVID-19, hypertension) where RAS is dysregulated. Ex vivo conditions may not fully replicate in vivo platelet behavior. The captopril-resistant ACE activity suggests a non-canonical form that warrants further investigation.

How to read the evidence

Well-designed ex vivo human platelet study with multiple validated assays. Negative result is well-supported by comprehensive testing across peptides and concentrations, though limited to healthy donors.

When this study was published

Published in 2025; addresses the ongoing question of RAS involvement in COVID-19 coagulopathy.

The bigger picture

The renin-angiotensin system has been extensively studied in the context of COVID-19 due to the virus using ACE2 for cell entry. This study helps clarify that while platelets express the molecular machinery of RAS, the system appears functionally inactive in healthy platelets, narrowing the search for mechanisms behind COVID-related clotting disorders.

Questions still open

  • Could RAS-platelet interactions become functionally relevant in disease states like COVID-19 or hypertension?
  • What is the captopril-resistant ACE-like activity detected in platelet lysates?
  • If RAS does not drive COVID-19 coagulopathy through platelets, what alternative pathways are responsible?

Common questions

What is the renin-angiotensin system and why was it studied in platelets?
The renin-angiotensin system (RAS) is a hormone system that regulates blood pressure through peptides like angiotensin II. Because COVID-19 uses ACE2 (a RAS component) to enter cells and causes abnormal blood clotting, researchers wanted to know if RAS peptides could directly activate platelets and cause clots.
Why is this negative result significant?
Negative results are valuable in science because they help eliminate incorrect hypotheses. By showing that angiotensin peptides do not activate healthy platelets despite receptor expression, this study redirects COVID-19 coagulopathy research toward more promising mechanisms.

Read the original research

The renin-angiotensin system in healthy human platelets: expressed but inactive.

Platelets, 36(1), 2546982

Citation

Panosetti, François; Cuenot, François M; Saint Auguste, Damian S; Martins Cavaco, Ana C; Nunes, Allancer D C; Lu, Philip H J; Magrini, Céline; Molot, Max; Sanglard, Gabriel; Günçü, Rodi; Zouaghi, Yassine; Béguelin, Charles; Martins Lima, Augusto; Stergiopulos, Nikolaos. (2025). The renin-angiotensin system in healthy human platelets: expressed but inactive.. Platelets, 36(1), 2546982. https://doi.org/10.1080/09537104.2025.2546982