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Study breakdown

GLP-1 Drug Exenatide Did Not Protect the Heart During Open-Heart Surgery in Large Clinical Trial

evidence
The takeaway

In a randomized trial of 1,389 patients, exenatide infusion during and after cardiopulmonary bypass surgery did not reduce death, stroke, kidney failure, or heart failure over nearly 6 years of follow-up.

24% vs. 24%

Identical rates of major adverse events in exenatide and placebo groups over nearly 6 years, definitively showing no perioperative cardioprotection.

What the researchers found

In this randomized, double-blind clinical trial of 1,389 predominantly low-risk patients undergoing elective coronary artery bypass grafting or aortic valve replacement:

- 170 patients (24%) in the exenatide group and 165 patients (24%) in the placebo group experienced the primary composite endpoint (death, stroke, renal failure requiring dialysis, or new/worsening heart failure)

- No significant difference in time to first event between groups

- No significant difference in rates of adverse events

- Median follow-up was 5.9 years (range 2.5–8.3 years)

- The study also tested liberal vs. restrictive oxygenation during bypass in a 2×2 factorial design, finding no difference there either (HR 1.0; 95% CI 0.83–1.3; p = 0.80)

Exenatide was administered as a 17.4 µg infusion during cardiopulmonary bypass and for the first hour after weaning from bypass.

Why it matters

This is an important negative result. While GLP-1 agonists have demonstrated cardiovascular benefits in diabetes and obesity trials, this study shows those benefits don't extend to acute perioperative cardioprotection during bypass surgery. This helps define the boundaries of GLP-1 drugs' cardiovascular effects and prevents unnecessary adoption of an ineffective intervention in cardiac surgery.

How the study worked

This was a randomized, double-blind, single-center clinical trial with a 2×2 factorial design. Adult patients undergoing elective cardiopulmonary bypass-assisted CABG or aortic valve replacement were randomized to receive either exenatide (17.4 µg infusion) or placebo during bypass and the first hour post-bypass, and to either liberal (100% FiO2) or restrictive (50% FiO2) oxygenation. The primary outcome was a composite of death, stroke, renal failure requiring dialysis, or new/worsening heart failure. Follow-up extended to a median of 5.9 years.

What this study cannot tell us

The study enrolled predominantly low-risk elective surgery patients, which may have limited the ability to detect benefit in a population with a low event rate. The exenatide infusion was given only during and briefly after bypass — a short exposure window that may be insufficient. Single-center design may limit generalizability. The 2×2 factorial design adds complexity to interpretation.

How to read the evidence

This is a large, well-designed randomized double-blind clinical trial with 1,389 patients and nearly 6 years of follow-up — high-quality evidence. The negative result is as informative as a positive one, establishing what GLP-1 agonists cannot do.

When this study was published

Published in 2025 with data from a trial registered in 2016 (NCT02673931). The long follow-up period (median 5.9 years) adds substantial value to the findings.

The bigger picture

GLP-1 agonists have shown cardiovascular benefits in the LEADER, SUSTAIN-6, and SELECT trials, raising hopes they could protect the heart in other settings. This trial tests the hypothesis in cardiac surgery and finds no benefit, suggesting that GLP-1's cardiovascular protection works through long-term metabolic and vascular mechanisms rather than acute cardioprotection during surgical ischemia-reperfusion injury.

Questions still open

  • Would longer perioperative GLP-1 agonist exposure (days rather than hours) provide cardioprotection in cardiac surgery?
  • Might GLP-1 agonists show benefit in higher-risk cardiac surgery patients with more room for improvement?
  • Does the lack of acute cardioprotection suggest GLP-1's cardiovascular benefits operate through chronic rather than acute mechanisms?

Common questions

If GLP-1 drugs protect the heart in other studies, why didn't exenatide work here?
The cardiovascular benefits of GLP-1 drugs seen in diabetes trials likely come from long-term effects on metabolism, blood vessels, and inflammation over months to years. Giving a single dose during surgery may be too brief to activate these protective mechanisms. The heart protection from GLP-1 drugs appears to be a chronic rather than acute effect.
Does this mean GLP-1 drugs aren't good for the heart?
No. Multiple large trials have shown that GLP-1 drugs reduce cardiovascular events when taken long-term for diabetes or obesity. This study specifically shows they don't provide additional protection when given as a brief infusion during heart surgery — a very different use case.

Read the original research

Efficacy of the Glucagon-Like Peptide-1 Agonist Exenatide in Patients Undergoing CABG or Aortic Valve Replacement: A Randomized Double-Blind Clinical Trial.

Circulation. Cardiovascular interventions, 18(5), e014961

Citation

Kjaergaard, Jesper; Møller, Christian Holdflod; Wiberg, Sebastian; Mikkelsen, Astrid Duus; Møller-Sørensen, Hasse; Ravn, Hanne Berg; Ravn, Jesper; Olsen, Peter Skov; Høfsten, Dan E; Boesgaard, Søren; Køber, Lars; Nilsson, Jens Christian; Hassager, Christian. (2025). Efficacy of the Glucagon-Like Peptide-1 Agonist Exenatide in Patients Undergoing CABG or Aortic Valve Replacement: A Randomized Double-Blind Clinical Trial.. Circulation. Cardiovascular interventions, 18(5), e014961. https://doi.org/10.1161/CIRCINTERVENTIONS.124.014961