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Structure-activity relationships of middle-size cyclic peptides, KRAS inhibitors derived from an mRNA display.

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Structure-activity relationships of middle-size cyclic peptides, KRAS inhibitors derived from an mRNA display.

Bioorganic & medicinal chemistry, 110, 117830

Citation

Kage, Mirai; Hayashi, Ryuji; Matsuo, Atsushi; Tamiya, Minoru; Kuramoto, Shino; Ohara, Kazuhiro; Irie, Machiko; Chiyoda, Aya; Takano, Koji; Ito, Toshiya; Kotake, Tomoya; Takeyama, Ryuuichi; Ishikawa, Shiho; Nomura, Kenichi; Furuichi, Noriyuki; Morita, Yuya; Hashimoto, Satoshi; Kawada, Hatsuo; Nishimura, Yoshikazu; Nii, Keiji; Sase, Hitoshi; Ohta, Atsushi; Kojima, Tetsuo; Iikura, Hitoshi; Tanada, Mikimasa; Shiraishi, Takuya. (2024). Structure-activity relationships of middle-size cyclic peptides, KRAS inhibitors derived from an mRNA display.. Bioorganic & medicinal chemistry, 110, 117830. https://doi.org/10.1016/j.bmc.2024.117830