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Study breakdown

Nociceptin Blocks ALL Three Types of Opioid Pain Relief in the Spinal Cord

Animal StudyPreliminary evidence
The takeaway

Nociceptin/orphanin FQ blocked antinociception induced by mu, kappa, AND delta opioid agonists at the spinal level, confirming it as a universal anti-opioid peptide that counteracts all forms of opioid-mediated pain relief.

Key finding

Nociceptin/OFQ blocked spinal antinociception from mu (DAMGO), kappa (U50,488H), and delta (DPDPE) opioid agonists in the cold water tail-flick test,

What the researchers found

Nociceptin/OFQ blocked spinal antinociception from mu (DAMGO), kappa (U50,488H), and delta (DPDPE) opioid agonists in the cold water tail-flick test, confirming nociceptin as a universal anti-opioid peptide opposing all three opioid receptor systems.

Why it matters

Relevant for opioid-peptides, neuropeptides, pain.

How the study worked

animal-study study on opioid-peptides, neuropeptides.

What this study cannot tell us

See abstract.

How to read the evidence

preliminary evidence.

When this study was published

Published in 2007.

The bigger picture

Advances peptide research.

Questions still open

  • Further research needed.
  • Clinical translation to evaluate.

Common questions

What was studied?
Nociceptin Blocks ALL Three Types of Opioid Pain Relief in the Spinal Cord
What was found?
Nociceptin/orphanin FQ blocked antinociception induced by mu, kappa, AND delta opioid agonists at the spinal level, confirming it as a universal anti-opioid peptide that counteracts all forms of opioid-mediated pain relief.

Read the original research

Nociceptin/orphanin FQ blocks the antinociception induced by mu, kappa and delta opioid agonists on the cold water tail-flick test.

European journal of pharmacology, 557(1), 32-6

Citation

Chen, Xiaohong; Geller, Ellen B; Adler, Martin W. (2007). Nociceptin/orphanin FQ blocks the antinociception induced by mu, kappa and delta opioid agonists on the cold water tail-flick test.. European journal of pharmacology, 557(1), 32-6.