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Study breakdown

Exenatide Did Not Reduce Heart Attacks or Amputations in Diabetic Patients With Peripheral Artery Disease

evidence
The takeaway

In the EXSCEL trial, diabetic patients with peripheral artery disease had higher mortality and amputation rates, but weekly exenatide did not improve cardiovascular events or amputation rates compared to placebo regardless of PAD status.

HR 1.38

Increased all-cause mortality in diabetic patients with PAD versus without PAD — highlighting the high-risk nature of this population

What the researchers found

Among 14,752 EXSCEL participants, 2,800 (19%) had PAD at baseline. PAD patients versus non-PAD patients had:

- Higher MACE rates: 13.6% vs 11.4% (adjusted HR 1.13, 95% CI 1.00-1.27, P=0.047)

- Higher all-cause mortality: adjusted HR 1.38 (95% CI 1.20-1.60, P<0.001)

- Higher LEA rates

Exenatide versus placebo showed no differences in MACE or lower-extremity amputation rates, regardless of PAD status. This means exenatide was neither beneficial nor harmful in this high-risk population.

Why it matters

Patients with both diabetes and PAD face extremely high cardiovascular risk and are at particular risk for lower-extremity amputation — a concern heightened after a diabetes drug (canagliflozin) was linked to increased amputation risk. This analysis provides safety reassurance that exenatide does not increase amputation risk in PAD patients. However, it also shows that exenatide does not provide the cardiovascular protection that newer GLP-1 agonists like semaglutide and liraglutide have demonstrated.

How the study worked

Post hoc analysis of the EXSCEL trial, a double-blind, placebo-controlled randomized trial evaluating once-weekly exenatide versus placebo in patients with type 2 diabetes. The primary endpoint was composite MACE (cardiovascular death, myocardial infarction, or stroke). This subgroup analysis assessed outcomes in patients with and without baseline PAD, with adjusted hazard ratios accounting for baseline characteristics.

What this study cannot tell us

This is a post hoc subgroup analysis, not a prespecified primary analysis, so it may be underpowered for detecting smaller treatment effects. PAD was defined by baseline medical history, which may undercount undiagnosed cases. Once-weekly exenatide is an older formulation; results may not apply to newer, more potent GLP-1 RAs. The null result for exenatide in PAD patients cannot be extrapolated to other GLP-1 drugs that have shown cardiovascular benefit.

How to read the evidence

This is a post hoc subgroup analysis from a large, well-conducted randomized controlled trial (EXSCEL, n=14,752). While the underlying trial is high-quality, post hoc analyses carry lower evidence strength than prespecified analyses.

When this study was published

Published in 2019 using EXSCEL trial data, this analysis predates the more recent cardiovascular outcome data for semaglutide and tirzepatide which have shown positive results.

The bigger picture

This analysis provides important context for understanding the heterogeneity of GLP-1 RA cardiovascular outcomes. While liraglutide (LEADER) and semaglutide (SUSTAIN-6) showed cardiovascular benefit, exenatide (EXSCEL) did not — and this subgroup analysis confirms the lack of benefit even in the highest-risk PAD population. This has contributed to the understanding that not all GLP-1 RAs are equivalent for cardiovascular protection, influencing guideline recommendations that favor specific agents.

Questions still open

  • Would semaglutide or liraglutide show cardiovascular benefit in the PAD subpopulation, given their overall positive CVOT results?
  • What explains the cardiovascular benefit heterogeneity among different GLP-1 receptor agonists?
  • Should GLP-1 RA selection for diabetic PAD patients prioritize agents with demonstrated cardiovascular benefit?

Common questions

Why was amputation risk specifically studied with this diabetes drug?
A different diabetes drug (canagliflozin, an SGLT2 inhibitor) was previously found to increase the risk of lower-extremity amputations in clinical trials, raising concerns about other diabetes medications. Since patients with peripheral artery disease already face high amputation risk, it was important to check whether exenatide had any effect on this outcome. Reassuringly, exenatide did not increase amputation risk.
If exenatide didn't help heart outcomes, does that mean GLP-1 drugs don't work for PAD patients?
Not necessarily. Exenatide is an older GLP-1 receptor agonist, and its overall EXSCEL trial was neutral for cardiovascular outcomes. Newer GLP-1 drugs — particularly semaglutide (SUSTAIN-6 trial) and liraglutide (LEADER trial) — have shown clear cardiovascular benefits. These newer agents may provide heart and vascular protection in PAD patients, though this would need to be confirmed in dedicated subgroup analyses.

Read the original research

Clinical Outcomes in Patients With Type 2 Diabetes Mellitus and Peripheral Artery Disease: Results From the EXSCEL Trial.

Circulation. Cardiovascular interventions, 12(12), e008018

Citation

Badjatiya, Anish; Merrill, Peter; Buse, John B; Goodman, Shaun G; Katona, Brian; Iqbal, Nayyar; Pagidipati, Neha J; Sattar, Naveed; Holman, Rury R; Hernandez, Adrian F; Mentz, Robert J; Patel, Manesh R; Jones, W Schuyler. (2019). Clinical Outcomes in Patients With Type 2 Diabetes Mellitus and Peripheral Artery Disease: Results From the EXSCEL Trial.. Circulation. Cardiovascular interventions, 12(12), e008018. https://doi.org/10.1161/CIRCINTERVENTIONS.119.008018