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Can Peptide-Targeted Radiation Therapy Treat Advanced Merkel Cell Skin Cancer? A Review of 37 Patients

evidence
The takeaway

In a review of 37 patients with metastatic Merkel cell carcinoma, peptide receptor radionuclide therapy (PRRT) produced objective responses in about 32% of cases with no severe side effects.

31.6% objective response rate

Six of 19 evaluable patients with metastatic Merkel cell carcinoma achieved partial or complete responses to PRRT with no severe adverse events.

What the researchers found

Of 37 patients with metastatic Merkel cell carcinoma who received 1-5 cycles of PRRT using 177Lu- or 90Y-labeled somatostatin analogs (cumulative activity 1.5-30 GBq), radiographic response data was available for 19 who received PRRT alone. Six of these 19 patients (31.6%) achieved objective responses ranging from partial to complete. No severe adverse events were reported across the treated cohort.

Why it matters

Metastatic Merkel cell carcinoma has limited treatment options and a poor prognosis. While immunotherapy has improved outcomes, many patients don't respond or eventually progress. PRRT offers a mechanistically different approach — using peptides to deliver targeted radiation directly to tumor cells — that could fill an important treatment gap for this rare cancer.

How the study worked

The authors performed a comprehensive literature review searching for all published reports of PRRT use in metastatic Merkel cell carcinoma. They compiled data from individual case reports and small series, totaling 37 treated patients. Response was assessed radiographically in patients who received PRRT as a standalone therapy.

What this study cannot tell us

The evidence quality is low — data comes from retrospective case reports and small series rather than controlled trials. The total of 37 patients is very small, and radiographic response data was only available for 19 who received PRRT alone. Publication bias likely favors positive outcomes. Patient selection (requiring somatostatin receptor expression) means results may not apply to all Merkel cell carcinoma cases.

How to read the evidence

This is a comprehensive literature review compiling data from case reports and small retrospective series. While it aggregates all available evidence, the underlying data quality is low — no randomized controlled trials exist yet. Prospective trials are underway.

When this study was published

Published in 2023, this review represents the most current synthesis of PRRT evidence for Merkel cell carcinoma as prospective trials begin enrolling.

The bigger picture

PRRT has already been approved for gastroenteropancreatic neuroendocrine tumors and is being explored for other cancers that express somatostatin receptors. Success in Merkel cell carcinoma would expand the reach of peptide-targeted radionuclide therapy to rare skin cancers. Prospective clinical trials are now underway to generate stronger evidence.

Questions still open

  • What proportion of Merkel cell carcinomas express sufficient somatostatin receptors for PRRT to be viable?
  • How does PRRT compare or combine with immunotherapy in this cancer type?
  • Will the ongoing prospective trials confirm the 32% response rate seen in this retrospective review?

Common questions

What is peptide receptor radionuclide therapy (PRRT)?
PRRT is a targeted cancer treatment that uses radioactive atoms attached to small peptides (somatostatin analogs). These peptides bind to specific receptors on tumor cells, delivering radiation directly to the cancer while minimizing damage to surrounding healthy tissue. It's already approved for certain neuroendocrine tumors.
Is PRRT effective for Merkel cell carcinoma?
Early evidence from 37 patients suggests PRRT may help — about 32% of evaluable patients showed tumor shrinkage with no severe side effects. However, the evidence comes from small retrospective studies, and prospective clinical trials are still needed to confirm these results. Only tumors that express somatostatin receptors are candidates for this therapy.

Read the original research

Peptide Receptor Radionuclide Therapy in Merkel Cell Carcinoma: A Comprehensive Review.

Journal of nuclear medicine technology, 51(1), 22-25

Citation

Askari, Emran; Moghadam, Soroush Zarehparvar; Wild, Damian; Delpassand, Ebrahim; Baldari, Sergio; Nilica, Bernhard; Hartrampf, Philipp E; Kong, Grace; Grana, Chiara Maria; Alexander Walter, Martin; Capoccetti, Francesca; Kasi, Pashtoon Murtaza; Strosberg, Jonathan. (2023). Peptide Receptor Radionuclide Therapy in Merkel Cell Carcinoma: A Comprehensive Review.. Journal of nuclear medicine technology, 51(1), 22-25. https://doi.org/10.2967/jnmt.122.264904